产品描述
A-674563 is an Akt1 inhibitor with Ki of 11 nM, modest potent to PKA and >30-fold selective for Akt1 over PKC
产品价格
货号 | 规格 | 价格 |
CC2826 |
2mg |
1036.00 元 |
CC2826 | 5mg | 1952.00 元 |
CC2826 | 10mg | 3463.00 元 |
化学数据
分子量Molecular Weight (MW) | 358.44 | |
---|---|---|
化学式Formula |
C22H22N4O |
|
CAS号CAS No. | 552325-73-2 | |
溶解性Solubility (25°C) | 二甲基亚砜DMSO |
72 mg/mL(200.87 mM) |
水Water | 72 mg/mL(200.87 mM) | |
乙醇Alcohol | 18 mg/mL(50.21 mM) |
制备储备液
浓度/溶剂体积(DMSO)/质量 | 1 mg | 5 mg | 10 mg |
1 mM | 2.7899 mL | 13.9493 mL | 27.8987 mL |
5 mM | 0.5580 mL | 2.7899 mL | 5.5797 mL |
10 mM | 0.2790 mL | 1.3949 mL | 2.7899 mL |
50 mM | 0.0558 mL | 0.2790 mL | 0.5580 mL |